Structural and thermodynamic basis of resistance to HIV-1 protease inhibition: Implications for inhibitor design

A. Velazquez-Campoy, S. Muzammil, H. Ohtaka, A. Schön, S. Vega, E. Freire. Structural and thermodynamic basis of resistance to HIV-1 protease inhibition: Implications for inhibitor design. Current Drug Targets: Infectious Disorders. 2003 3:311-328